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Metabolism Alprazolam is extensively metabolized in people, generally by cytochrome P450 3A4 (CYP3A4), to 2 main active metabolites within the plasma: four-hydroxyalprazolam and α-hydroxyalprazolam. The plasma circulation levels of The 2 active metabolites are less than 4% with the dad or mum. The noted relative potencies in benzodiazepine recepto